发明名称 |
AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME |
摘要 |
New aminoacid derivates have the general formula: T-Z-NR<1>-(R<2>CR<3>)-CO-Y-(CH2)n-R, in which R, R<1> to R<3>, T, Z, Y and n are defined as in the first claim. They represent valuable NPY-antagonistic active substances. Also disclosed are their diastereomers, their enantiomers and their salts, in particular their physiologically tolerable salts with inorganic or organic acids or bases, as well as medicaments containing these compounds, their use and a process for preparing the same. |
申请公布号 |
WO9417035(A1) |
申请公布日期 |
1994.08.04 |
申请号 |
WO1994EP00109 |
申请日期 |
1994.01.18 |
申请人 |
DR. KARL THOMAE GMBH |
发明人 |
RUDOLF, KLAUS;EBERLEIN, WOLFGANG;ENGEL, WOLFHARD;MIHM, GERHARD;DOODS, HENRI;WIELAND, HEIKE-ANDREA;WILLIM, KLAUS-DIETER;KRAUSE, JUERGEN;DOLLINGER, HORST;ESSER, FRANZ;SCHNORRENBERG, GERD;ENTZEROTH, MICHAEL;WIENEN, WOLFGANG |
分类号 |
A61K31/155;A61K31/165;A61K31/195;A61K31/198;A61K31/38;A61K31/381;A61K31/40;A61K31/403;A61K31/404;A61K31/41;A61K31/415;A61K31/4184;A61K31/4245;A61K31/44;A61K31/4409;A61K31/4418;A61K31/4427;A61K31/445;A61K31/4465;A61K31/4468;A61K31/454;A61K31/47;A61K38/00;A61P9/12;A61P43/00;C07C237/22;C07C237/42;C07C255/60;C07C257/12;C07C257/14;C07C257/18;C07C259/10;C07C259/18;C07C261/04;C07C275/40;C07C279/10;C07C279/12;C07C279/14;C07C279/18;C07C279/36;C07C307/02;C07C307/10;C07C311/08;C07C311/15;C07C311/19;C07C311/39;C07C311/42;C07D209/14;C07D209/16;C07D209/42;C07D209/44;C07D211/28;C07D213/38;C07D213/55;C07D215/12;C07D215/38;C07D223/20;C07D233/24;C07D233/48;C07D233/54;C07D233/64;C07D233/66;C07D233/72;C07D233/88;C07D235/06;C07D235/08;C07D249/08;C07D249/10;C07D249/12;C07D249/14;C07D271/06;C07D271/07;C07D295/15;C07D333/20;C07D333/36;C07D401/12;C07D471/04;C07K5/072;(IPC1-7):C07C279/14 |
主分类号 |
A61K31/155 |
代理机构 |
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