发明名称 Chemical process
摘要 A process for the preparation of a 5,7-diaryloxy-2-(2-heteroaryl)-triazolo[1,5-a][1,3,5]triazine, which comprises reacting a N-2-(4,6-diaryloxy)-[1,3,5]triazinyl-N'-(2-heteroarylcarbonyl)hydrazine with a polyphosphoric acid silyl ester. The invention also provides a multistep process for preparing certain triazolotriazines having activity asadenosine antagonists.
申请公布号 US5326869(A) 申请公布日期 1994.07.05
申请号 US19920979096 申请日期 1992.11.20
申请人 IMPERIAL CHEMICAL INDUSTRIES, PLC 发明人 HUTTON, JONATHAN
分类号 A61K31/53;A61P9/00;A61P9/10;A61P25/04;A61P25/06;C07D487/04;C07D513/04;(IPC1-7):C07D487/04 主分类号 A61K31/53
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