发明名称 |
Substituted pyrimidines, pyrimidinones and pyridopyrimidines |
摘要 |
Substituted pyrimidines, pyrimidinones and pyridopyrimidines of formula (I) are as angiotensin II antagonists useful in the treatment of hypertension, ocular hypertension and certain CNS ailments: <IMAGE> (I) wherein K is -N(R8a)-C(=M) or -N=C(R8b) where M is O or NR22.
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申请公布号 |
US5324729(A) |
申请公布日期 |
1994.06.28 |
申请号 |
US19920908143 |
申请日期 |
1992.07.31 |
申请人 |
MERCK & CO., INC. |
发明人 |
ALLEN, ERIC E.;GREENLEE, WILLIAM J.;MACCOSS, MALCOLM;PATCHETT, ARTHUR A. |
分类号 |
C07D239/26;C07D239/28;C07D239/36;C07D239/38;C07D239/42;C07D403/10;C07D471/04;C07F9/6512;(IPC1-7):C07D471/04;A61K31/505 |
主分类号 |
C07D239/26 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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