发明名称 Optically active 5-oxygenated (3S)-1,3-dimethyloxindole-3-acetic acids
摘要 The synthesis of optically active 5-oxygenated (3S)-1,3-dimethyloxindole-3-acetic acids R = H, CH3, C2H5, CH2Ph <IMAGE> R = H, CH3, C2H5, CH2Ph and their use in the synthesis of optically active (3aS-cis)-eseroline and (3aS-cis)-N1-benzylnoreseroline, which are important intermediates in the synthesis of compounds related to (3aS-cis)-physostigmine and carbamate analogs, and of (3aS-cis)-N1-benzylnor- and N1-norphysostigmine and their carbamate analogs.
申请公布号 US5310935(A) 申请公布日期 1994.05.10
申请号 US19920906508 申请日期 1992.06.30
申请人 PHARMAGROUP INTERNATIONAL 发明人 BROSSI, ARNOLD;MASSARI, DANILO C.;YU, QIAN-SHENG
分类号 C07D209/34;C07D487/04;C07D491/04;(IPC1-7):C07D209/34 主分类号 C07D209/34
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