发明名称 Azole compound
摘要 A compound represented by general formula (I), wherein R<1> represents imidazolyl, triazolyl or tetrazolyl each of which may be substituted by methyl and/or ethyl. R<2> represents naphthyl, phenanthryl or anthryl each of which may be substituted by substituent(s) selected from the following group A: C1-C4 alkyl, C1-C4 alkoxy, C1-C6 acyloxy, aromatic acyloxy, OH, trialkyl, C1-C4 acyl amino, alkoxyalkoxy, alkoxyacyloxy and trialkylsilyloxy; and R<3> represents hydrogen, methyl or cyano. This compound has an excellent aromatase inhibitor activity and is useful particularly as a remedy for breast cancer.
申请公布号 AU5285593(A) 申请公布日期 1994.05.09
申请号 AU19930052855 申请日期 1993.10.20
申请人 SANKYO COMPANY, LIMITED 发明人 TOMOYUKI SHIBATA;YUKIO SUGIMURA;KAZUHIKO TANZAWA;MASAAKI TAKAHASHI;TOMOWO KOBAYASHI;YOSHIHIRO MITSUHASHI
分类号 C07D233/54;C07D233/61;C07D233/64;C07D257/04;C07D521/00 主分类号 C07D233/54
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