发明名称 O-ALKYLATED RAPAMYCIN DERIVATIVES AND THEIR USE, PARTICULARLY AS IMMUNOSUPPRESSANTS
摘要 Novel O-alkylated derivatives of rapamycin of formula (I), especially 40-O-alkylated derivatives, are found to have pharmaceutical utility, particularly as immunosuppressants.
申请公布号 WO9409010(A1) 申请公布日期 1994.04.28
申请号 WO1993EP02604 申请日期 1993.09.24
申请人 SANDOZ-ERFINDUNGEN VERWALTUNGSGESELLSCHAFT M.B.H.;SANDOZ-PATENT-GMBH;SANDOZ LTD. 发明人 COTTENS, SYLVAIN;SEDRANI, RICHARD
分类号 A61K31/00;A61K31/435;A61K31/4353;A61K31/436;A61K31/455;A61K31/496;A61K31/52;A61K31/5377;A61K31/573;A61K38/00;A61K39/395;A61P11/00;A61P11/06;A61P29/00;A61P31/00;A61P31/04;A61P35/00;A61P35/02;A61P37/00;A61P37/06;A61P43/00;C07D498/18;C07F7/18;(IPC1-7):C07D498/18 主分类号 A61K31/00
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