发明名称 |
Tetrahydro 2-saccharinylmerthyl aryl carboxylates |
摘要 |
4-R4-R5-Saccharinylmethyl aryl carboxylates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R4-R5-2-halomethylsaccharin with an arylcarboxylic acid in the presence of an acid-acceptor.
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申请公布号 |
US5306818(A) |
申请公布日期 |
1994.04.26 |
申请号 |
US19920965593 |
申请日期 |
1992.10.23 |
申请人 |
STERLING WINTHROP INC. |
发明人 |
SUBRAMANYAM, CHAKRAPANI;BELL, MALCOLM R. |
分类号 |
A61K31/425;A61K31/435;A61P1/00;A61P11/00;A61P29/00;A61P43/00;C07D275/06;C07D413/12;C07D417/04;C07D417/12;C07F9/6541;(IPC1-7):C07D275/06 |
主分类号 |
A61K31/425 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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