发明名称 SUBSTITUTED ACETAMIDE DERIVATIVES
摘要 There are provided substituted acetamide derivatives represented by general formula (I): (I) wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11, R12, R13, n and Z are defined in the specification. The substituted acetamide derivatives strongly inhibit acylcoenzyme A cholesterol acyltransferase (ACTA) and are expected to be effective for the treatment and prevention of hypercholesterolemia, hyperlipemia and arteriosclerosis.
申请公布号 CA2105617(A1) 申请公布日期 1994.03.11
申请号 CA19932105617 申请日期 1993.09.07
申请人 BANYU PHARMACEUTICAL CO., LTD. 发明人 IWASAWA, YOSHIKAZU;HATTORI, HIROMI;NAGATA, YASUFUMI;SHIMIZU, AKIKO;SAWASAKI, YOSHIO
分类号 C07C317/44;C07C323/60;C07D215/36;C07D233/28;C07D233/84;C07D239/38;C07D307/91;C07D333/18;(IPC1-7):C07C323/41;A61K31/165;C07C317/32;A61K31/33;C07D277/36;C07D263/46;C07D333/62;C07D213/70 主分类号 C07C317/44
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