发明名称 IMIDAZOLE DERIVATIVES
摘要 Novel 4,5-dicyanoimidazole derivatives of formula (I), wherein X is oxygen, sulfur, SO or SO2; R1 is hydrogen, C1-C6alkyl, C1--C6haloalkyl, C1-C6hydroxyalkyl, C1-C6cyanoalkyl, or a C1-C6alkylene substituted by C1-C6alkoxy, C1-C6haloalkoxy, C1-C6alkylthio, C1-C6haloalkylthio, C1-C6alkylsulfinyl, C1-C6haloalkylsulfinyl, C1-C6alkylsulfonyl, C1-C6haloalkylsulfonyl, C1-C6hydroxyalkyl, C1-C6alkyloxycarbonyl, C1-C6alkylcarbonyl, C1-C6alkylcarbonyloxy or by COOH; R2 is hydrogen, halogen, CN, C1-C6alkyl, C1-C6haloalkyl, C1-C6cyanoalkyl, C1-C6hydroxyalkyl, C1-C6alkoxy, C1-C6haloalkoxy, C1-C6alkylthio, C1-C6haloalkylthio or C3-C7cycloalkyl; R3 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, cyano or nitro; R4 is hydrogen, halogen, nitro, cyano, NCS, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; and R5 is hydrogen, halogen, nitro, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; or R4 and R5 together form a -O-(CH2)m-O- bridge, wherein m is an integer selected from the group consisting of 1, 2 and 3, with the proviso that R4 and R5 are located at adjacent carbon atoms; including the physiologically tolerable addition compounds, can be used against insects and representatives of the order Acarina that are harmful to animals and plants, as well as against helminths in warm-blooded animals.
申请公布号 WO9401432(A1) 申请公布日期 1994.01.20
申请号 WO1993EP01682 申请日期 1993.06.30
申请人 CIBA-GEIGY AG 发明人 HILDENBRAND, CHRISTOF;GEHRET, JEAN-CLAUDE;TINEMBART, OLIVIER
分类号 A01N43/78;A61K31/425;A61P33/10;C07D417/12;C07D513/04;(IPC1-7):C07D417/12;C07D277/68;C07D277/74;C07D277/76 主分类号 A01N43/78
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