发明名称 Process for preparation of beta-lactam derivatives.
摘要 <p>The invention provides a process for preparing a beta -lactam derivative represented by the formula <CHEM> the process comprising reacting a beta -lactam derivative represented by the following formula (II) and having a protected carboxyl group with a cresol; <CHEM> wherein R represents a benzyl group having an electron-donating group as a substituent on the phenyl ring, a diphenylmethyl group which may have an electron-donating group as a substituent on the phenyl ring or a tert-butyl group.</p>
申请公布号 EP0331146(B1) 申请公布日期 1994.01.12
申请号 EP19890103587 申请日期 1989.03.01
申请人 OTSUKA KAGAKU KABUSHIKI KAISHA;TAIHO PHARMACEUTICAL COMPANY LIMITED 发明人 TANIGUCHI, MASATOSHI;SASAOKA, MICHIO;MATSUMURA, KIYOTOSHI;KAWAHARA, ICHIRO;KAZE, KENJI;SUZUKI, DAISUKE;SHIMABAYASHI, AKIHIRO
分类号 C07D499/87;C07D499/00;C07D499/08;C07D499/86;C07D499/897;(IPC1-7):C07D499/00 主分类号 C07D499/87
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