发明名称 Hydroxy-4-benzenethio derivatives, their preparation as well as their use for the preparation of aminoalkoxybenzenesulfonyle derivatives.
摘要 <p>The subject of the invention is 4-hydroxybenzenethio (4-hydroxyphenylthio) derivatives of general formula &lt;IMAGE&gt; in which: R1 and R2, which are identical or different, each represent hydrogen, the methyl or ethyl radical or a halogen atom, R represents a C1-C6 alkyl, C3-C6 cycloalkyl or phenyl radical, R3 represents hydrogen or a halogen atom, X represents -O-, -S- or &lt;IMAGE&gt; in which R4 represents hydrogen or a C1-C4 alkyl group, useful as synthetic intermediates, especially for the preparation of aminoalkoxybenzenesulphonyl (aminoalkoxyphenylsulphonyl) derivatives which are pharmaceutically active compounds.</p>
申请公布号 EP0576347(A1) 申请公布日期 1993.12.29
申请号 EP19930401600 申请日期 1993.06.22
申请人 ELF SANOFI 发明人 GUBIN, JEAN;INION, HENRI
分类号 C07D209/30;C07D307/82;C07D333/62;C07D403/12;C07D405/12;C07D409/12;(IPC1-7):C07D209/30 主分类号 C07D209/30
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