发明名称 |
NEW DELTA-17 AND DELTA-20 OLEFINIC AND SATURATED 17 beta -SUBSTITUTED-4-AZA-5 alpha -ANDROSTAN-3-ONES AS 5 alpha -REDUCTASE INHIBITORS |
摘要 |
Described are new delta-17 and delta-20 olefinic and saturated 17 beta -substituted 4-aza-5 alpha -androstan-3-ones and related compounds and the use of such compounds as 5 alpha -reductase inhibitors for treatment of benign prostatic hyperplasia and other hyperandrogenic related disorders. |
申请公布号 |
WO9323050(A1) |
申请公布日期 |
1993.11.25 |
申请号 |
WO1993US04630 |
申请日期 |
1993.05.17 |
申请人 |
MERCK & CO., INC. |
发明人 |
GRAHAM, DONALD, W.;ASTER, SUSAN, D.;TOLMAN, RICHARD, L. |
分类号 |
A61K8/63;A61K8/00;A61K31/58;A61Q5/00;A61Q7/00;A61Q19/00;C07J73/00;(IPC1-7):A61K31/495;C07D241/02 |
主分类号 |
A61K8/63 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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