发明名称 NEW DELTA-17 AND DELTA-20 OLEFINIC AND SATURATED 17 beta -SUBSTITUTED-4-AZA-5 alpha -ANDROSTAN-3-ONES AS 5 alpha -REDUCTASE INHIBITORS
摘要 Described are new delta-17 and delta-20 olefinic and saturated 17 beta -substituted 4-aza-5 alpha -androstan-3-ones and related compounds and the use of such compounds as 5 alpha -reductase inhibitors for treatment of benign prostatic hyperplasia and other hyperandrogenic related disorders.
申请公布号 WO9323050(A1) 申请公布日期 1993.11.25
申请号 WO1993US04630 申请日期 1993.05.17
申请人 MERCK & CO., INC. 发明人 GRAHAM, DONALD, W.;ASTER, SUSAN, D.;TOLMAN, RICHARD, L.
分类号 A61K8/63;A61K8/00;A61K31/58;A61Q5/00;A61Q7/00;A61Q19/00;C07J73/00;(IPC1-7):A61K31/495;C07D241/02 主分类号 A61K8/63
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