| 摘要 |
3-(Indole-2-carboxamido)quinuclidines of the formula 1 Ind-CO-NHR in which Ind denotes a 2-indolyl group which is unsubstituted or mono- to trisubstituted by alkyl, alkoxy, alkoxycarbonyl and/or alkylthio each having 1-4 C atoms, 7-11 C-aralkyloxy, 1-5 C-acyloxy, 6-10 C-aroyloxy, 6-10 C-aryloxy, trifluoromethyl, cyano, fluorine, chlorine, hydroxyl, 1-4 C-alkylsulphonyloxy, 6-10 C-arylsulphonyloxy, carboxyl and/or methylenedioxy and R denotes 3-quinuclidinyl and their physiologically acceptable salts, which show selective serotonin-antagonistic action and can be used as psychopharmaceuticals. |
