发明名称 Certain 9-amino-2-(or 4)-oxa 1,2,3,4-tetrahydro- or 1,2,3,4,5,6,7,8-octahydro-acridines
摘要 PCT No. PCT/US88/01070 Sec. 371 Date Apr. 27, 1990 Sec. 102(e) Date Apr. 27, 1990 PCT Filed Mar. 30, 1988 PCT Pub. No. WO89/02740 PCT Pub. Date Apr. 6, 1989.Compounds selected from the group consisting of 9-amino-4-oxa-1,2,3,4-tetrahydro-acridine, 9-amino-2-oxa-1,2,3,4-tetrahydro-acridine, 9-amino-8-fluoro-4-oxa-1,2,3,4-tetrahydro-acridine, 9-amino-4-oxa-1,2,3,4,5,6,7,8-octahydro-acridine or a pharmaceutical acceptable salt thereof are useful treating Alzheimer's disease.
申请公布号 US5202440(A) 申请公布日期 1993.04.13
申请号 US19900474717 申请日期 1990.04.27
申请人 PFIZER INC. 发明人 DESAI, MANOJ C.
分类号 C07C255/61;C07D213/84;C07D213/85;C07D219/10;C07D221/16;C07D221/22;C07D307/30;C07D309/28;C07D311/68;C07D333/36;C07D335/02;C07D335/06;C07D405/12;C07D471/04;C07D491/04;C07D491/052;C07D491/14;C07D495/04;C07D495/14;C07D498/04;C07D513/04 主分类号 C07C255/61
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