发明名称 |
AZELASTIN ENTHALTENDE ARZNEIMITTEL ZUR ANWENDUNG IN DER NASE UND/ODER AM AUGE. |
摘要 |
Medicaments for nasal or ocular admin. contain 0.0005-2 wt% of azelastin (I) or its salts. (I) is 4-(4-chlorobenzyl)-2 (perhydro-1-methyl-4-azepinyl) -1(2H)-phthalazinone and is described in DE 2164058 (as an antiallergic agent). The medicaments are formulated as aq. solns., gels, ointments, aerosol suspensions or powders. Solns. contain 0.001-0.1% of a preservative, esp. thiomersal or an alkyl benzyl diemthyl ammonium chloride, and may also contain up to 15% of a water-miscible solvent.
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申请公布号 |
DE3877904(D1) |
申请公布日期 |
1993.03.11 |
申请号 |
DE19883877904 |
申请日期 |
1988.10.27 |
申请人 |
ASTA PHARMA AG, 6000 FRANKFURT, DE |
发明人 |
HETTCHE, DR., HELMUT, W-6057 DIETZENBACH, DE |
分类号 |
A61K9/06;A61K31/55;(IPC1-7):A61K31/55 |
主分类号 |
A61K9/06 |
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