发明名称 2-(PYRROLIDINYL-1-METHYL)-PIPERIDINE DERIVATIVES AND THEIR USE AS KAPPA-RECEPT OR AGONISTS
摘要 Azacyclic derivatives of formula (I), are kappa-receptor agonists and are useful in the treatment of convulsions, cough, asthma, inflammation, pancreatitis, arrhythmias, hyponatraemic disease states and cerebral ischaemia.
申请公布号 AU1760992(A) 申请公布日期 1992.12.30
申请号 AU19920017609 申请日期 1992.05.15
申请人 DR LO ZAMBELETTI S.P.A. 发明人 GIUSEPPE GIARDINA;ROBERTO COLLE;GEOFFREY DOUGLAS CLARKE
分类号 A61K31/445;A61K31/4427;A61P7/10;A61P9/06;A61P9/10;A61P11/00;A61P25/02;A61P25/08;A61P25/28;A61P29/00;C07D401/06 主分类号 A61K31/445
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