发明名称 |
Steroid esters of methylated prostaglandin derivatives and their pharmaceutical compositions. |
摘要 |
<p>Methylated prostaglandine derivatives are steroid derivatives having at 17 position, methylated prostaglandine group such as
<UnorderedLists id="ula01" listStyle="none"><ListItem>(Me)<Sub>2</Sub>-PGE<Sub>2</Sub>-E</ListItem><ListItem>(Me)<Sub>2</Sub>-PGE<Sub>2</Sub>-E-2AC</ListItem><ListItem>(Me)<Sub>2</Sub>-PGE<Sub>2</Sub>-E-BA</ListItem><ListItem>(Me)<Sub>2</Sub>-PGE<Sub>2</Sub>-E-2AC-BA</ListItem><ListItem>(Me)-PGF<Sub>2</Sub>a-E</ListItem><ListItem>(Me)-PGF<Sub>2</Sub>a-E-3AC</ListItem><ListItem>(Me)-PGF<Sub>2</Sub>a-E-BA or</ListItem><ListItem>(Me)-PGF<Sub>2</Sub>a-E-3AC-BA</ListItem></UnorderedLists></p><p>or 600 mg/kg of the following active ingredient:
<UnorderedLists id="ula02" listStyle="none"><ListItem>(Me)<Sub>2</Sub>-PGE<Sub>2</Sub>'-E</ListItem><ListItem>(Me)<Sub>2</Sub>-PGE<Sub>2</Sub>'-E-2AC</ListItem><ListItem>(Me)<Sub>2</Sub>-PGE<Sub>2</Sub>'-E-BA</ListItem><ListItem>(Me)<Sub>2</Sub>-PGE<Sub>2</Sub>'-E-2AC-BA</ListItem><ListItem>(Me)-PGE<Sub>2</Sub>-E</ListItem><ListItem>(Me)-PGE<Sub>2</Sub>-E-2AC</ListItem><ListItem>(Me)-PGE<Sub>2</Sub>-E-BA or</ListItem><ListItem>(Me)-PGE<Sub>2</Sub>-E-2AC-BA.</ListItem></UnorderedLists></p> |
申请公布号 |
EP0030299(A1) |
申请公布日期 |
1981.06.17 |
申请号 |
EP19800107209 |
申请日期 |
1980.11.19 |
申请人 |
KUREHA KAGAKU KOGYO KABUSHIKI KAISHA |
发明人 |
ENOMOTO, SATORU;ASANO, KIRO;TAMURA, HUMIO;TANAKA, HIROMITSU |
分类号 |
C07C405/00;C07J1/00;(IPC1-7):07C177/00;07J1/00;07J5/00;07J71/00 |
主分类号 |
C07C405/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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