发明名称 |
NOVEL HETEROCYCLIC CARBOXYLIC ACIDS |
摘要 |
The present invention relates to novel N-substituted azaheterocyclic carboxylic acids and esters thereof of formula (I), a method of preparing the same and to pharmaceutical compositions comprising the compounds. The novel compounds are useful in treating a central nervous system ailment related to the GABA uptake. Compounds of formula (I) may be used to treat for example, pain, anxiety, extrapyrimidinal dyskinesia, epilepsy and certain muscular and movement disorders. They are also useful as sedatives, hypnotics and antidepressants. |
申请公布号 |
WO9220658(A1) |
申请公布日期 |
1992.11.26 |
申请号 |
WO1992DK00155 |
申请日期 |
1992.05.14 |
申请人 |
NOVO NORDISK A/S |
发明人 |
ANDERSEN, KNUD, ERIK;KNUTSEN, LARS, JACOB, STRAY;SOERENSEN, PER, OLAV;LUNDT, BEHREND, FRIEDRICH;LAU, JESPER;PETERSEN, HANS |
分类号 |
A61K31/395;A61K31/4427;A61K31/445;A61K31/455;A61K31/54;A61K31/5415;A61K31/55;A61K31/554;A61P25/04;A61P25/08;A61P25/20;A61P25/24;A61P25/26;C07D207/08;C07D207/16;C07D211/36;C07D211/60;C07D279/22;C07D281/02;C07D281/16;C07D281/18;C07D335/10;C07D337/14;C07D337/16;C07D401/06;C07D401/12;C07D403/12;C07D413/12;C07D417/12 |
主分类号 |
A61K31/395 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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