发明名称 |
Benzodiazepine derivatives, compositions containing them and their use in therapy. |
摘要 |
<p>Compounds of formula (I), and salts and prodrugs thereof <CHEM> wherein: R<1> represents optionally substituted C1-6alkyl or C3-7cycloalkyl; R<2> represents an optionally substituted phenyl or pyridyl group; R<3> represents C1-6 alkyl or halo; R<4> represents C3-7 cycloalkyl; X is 0, 1, 2 or 3; are CCK and/or gastrin antagonists. They and compositions thereof are therefore useful in therapy.</p> |
申请公布号 |
EP0514133(A1) |
申请公布日期 |
1992.11.19 |
申请号 |
EP19920304264 |
申请日期 |
1992.05.12 |
申请人 |
MERCK SHARP & DOHME LTD. |
发明人 |
CHAMBERS, MARK S.;FLETCHER, STEPHEN R.;MATASSA, VICTOR G. |
分类号 |
A61K31/55;A61K31/551;A61P1/00;A61P1/04;A61P3/04;A61P25/00;A61P25/02;C07D243/14;C07D243/24;C07D401/12;C07D403/12;C07D417/12;C07D521/00 |
主分类号 |
A61K31/55 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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