发明名称 Benzodiazepine derivatives, compositions containing them and their use in therapy.
摘要 <p>Compounds of formula (I), and salts and prodrugs thereof &lt;CHEM&gt; wherein: R&lt;1&gt; represents optionally substituted C1-6alkyl or C3-7cycloalkyl; R&lt;2&gt; represents an optionally substituted phenyl or pyridyl group; R&lt;3&gt; represents C1-6 alkyl or halo; R&lt;4&gt; represents C3-7 cycloalkyl; X is 0, 1, 2 or 3; are CCK and/or gastrin antagonists. They and compositions thereof are therefore useful in therapy.</p>
申请公布号 EP0514133(A1) 申请公布日期 1992.11.19
申请号 EP19920304264 申请日期 1992.05.12
申请人 MERCK SHARP & DOHME LTD. 发明人 CHAMBERS, MARK S.;FLETCHER, STEPHEN R.;MATASSA, VICTOR G.
分类号 A61K31/55;A61K31/551;A61P1/00;A61P1/04;A61P3/04;A61P25/00;A61P25/02;C07D243/14;C07D243/24;C07D401/12;C07D403/12;C07D417/12;C07D521/00 主分类号 A61K31/55
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