发明名称 |
2,4-AND 2,5-BISTETRAZOLYLPYRIDINES,A PROCESS FOR THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICALS |
摘要 |
The invention relates to 2,4- and 2,5-bis(tetrazolyl)pyridines. The said compounds inhibit the enzymes proline hydroxylase and lysine hydroxylase and cause selective inhibition of collagen biosynthesis. They are used as fibrosuppressants and immunosuppresants. |
申请公布号 |
ZA9200788(B) |
申请公布日期 |
1992.10.28 |
申请号 |
ZA19920000788 |
申请日期 |
1992.02.04 |
申请人 |
HOECHST AKTIENGESELLSCHAFT |
发明人 |
GERRIT SCHUBERT;EKKEHARD BAADER;MARTIN BICKEL;VOLKMAR GUENZLER-PUKALL |
分类号 |
A61K31/44;A61K31/4409;A61K31/4427;A61P7/02;A61P37/06;A61P43/00;C07D213/04;C07D257/04;C07D401/04;C07D401/14;C07D405/14 |
主分类号 |
A61K31/44 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|