| 发明名称 |
PYRROLIDINYLAMIDE ESTER DERIVATIVE HAVING ANTI-PROLYL ENDOPEPTIDASE ACTIVITY, ITS SYNTHESIS AND USE AND A PHARMACEUTICAL COMPOSITION CONTAINING IT |
| 摘要 |
<p>A novel pyrrolidinylamide ester derivative that exhibits inhibitory activity against prolyl endopeptidase, methods for synthesis thereof and its use as an inhibitor against said enzyme are disclosed. The pyrrolidinylamide ester of the invention has the following general formula: <IMAGE> wherein n is 0 or an integer of 1 to 7 and R is hydrogen atom or a straight or branched alkyl having 1 to 8 carbon atoms.</p> |
| 申请公布号 |
GR3001441(T3) |
申请公布日期 |
1992.09.25 |
| 申请号 |
GR19900400720T |
申请日期 |
1991.02.07 |
| 申请人 |
SUNTORY LIMITED |
发明人 |
HIGUCHI, NAOKI;SAITOH, MASAYUKI;HASHIMOTO, MASAKI;FUKAMI, HARUKAZU 15-1-709, KUJO-CHO KISSHOIN;TANAKA, TAKAHARU 1-5-1-801, HIGASHIAWAJI |
| 分类号 |
A61K31/445;A61K31/40;A61K31/401;A61P25/00;A61P43/00;C07D295/10;C07D295/185;C12N9/99;(IPC1-7):C07D295/18 |
主分类号 |
A61K31/445 |
| 代理机构 |
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