ALDOPHOSPHAMIDE GLYCOSIDES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICAL ACTIVE COMPOUNDS

摘要

Compounds of the formula <IMAGE> (I) <IMAGE> or <IMAGE> (III) in which R1 represents saturated, unsaturated or anhydro desoxypentosyl, desoxyhexosyl or didesoxyhexosyl, where the OH functions of the sugar are optionally protected, and R2 represents straight-chain or branched or heterosubstituted alkyl having up to ten carbon atoms and R3 represents straight-chain or branched or heterosubstituted alkyl having up to ten carbon atoms and X represents halogens and R4 represents straight-chain or branched or heterosubstituted alkyl having up to ten carbon atoms. Such compounds are useful as highly selective cytostatics in cancer therapy.