| 发明名称 |
2,6-METHANO-2H-1-BENZOXOCINCARBOXAMIDES AS 5-HT3-ANTAGONISTS |
| 摘要 |
Novel compounds which are 2,6-methano-2H-1-benzoxocincarboxamides having 5-HT3-antagonist properties including unique CNS, anti-emetic and gastric prokinetic activities and which are void of any significant D2 receptor binding affinity, processes for their preparation, therapeutic compositions and methods of treatment of disorders which result from 5-HT3 activity using said compounds are disclosed. |
| 申请公布号 |
AU9102991(A) |
申请公布日期 |
1992.06.25 |
| 申请号 |
AU19910091029 |
申请日期 |
1991.11.22 |
| 申请人 |
RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. |
发明人 |
JOHN E AIREY;MATTHEW R POWERS;WALTER RODRIGUEZ;RAYMOND D. YOUSSEFYEH |
| 分类号 |
C07D313/20;C07D453/02;(IPC1-7):A61K31/55;A61K31/435;A61K31/445;C07D451/14;A61K31/535;C07D405/12;C07D471/08;C07D498/08;C07D513/08 |
主分类号 |
C07D313/20 |
| 代理机构 |
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