发明名称 RETROVIRAL PROTEASE INHIBITORS
摘要 Compounds represented by formula (I), wherein A represents R, R<13> and radicals represented by formulas (A1, A2, A3), B represents radicals represented by formula (II), (values for the variables given herein), are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease.
申请公布号 WO9208688(A1) 申请公布日期 1992.05.29
申请号 WO1991US08617 申请日期 1991.11.18
申请人 MONSANTO COMPANY 发明人 BERTENSHAW, DEBORAH, ELIZABETH;FRESKOS, JOHN, NICHOLAS;GETMAN, DANIEL, PAUL;HEINTZ, ROBERT, MARTIN;LIN, KO-CHUNG;ROGIER, DONALD, JOSEPH, JR.;TALLEY, JOHN, JEFFREY
分类号 A61K31/17;A61K31/185;A61K31/195;A61K31/197;A61K31/216;A61K31/27;A61K31/34;A61K31/343;A61K31/40;A61K31/415;A61K31/4184;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4418;A61K31/4427;A61K31/445;A61K31/454;A61K31/47;A61K31/4709;A61K31/472;A61K31/496;A61K31/505;A61K31/535;A61K31/5355;A61K31/5375;A61K31/5377;A61K38/00;A61P31/12;A61P37/04;A61P43/00;C07C69/593;C07C213/00;C07C213/02;C07C213/08;C07C215/28;C07C271/16;C07C271/20;C07C271/22;C07C275/04;C07C275/14;C07C275/18;C07C275/22;C07C275/24;C07C275/26;C07C275/28;C07C275/40;C07C311/31;C07C311/45;C07C311/47;C07C317/28;C07C317/40;C07C317/44;C07C317/48;C07C317/50;C07C323/40;C07C323/60;C07C329/06;C07C335/08;C07C335/12;C07D207/16;C07D211/16;C07D213/40;C07D213/81;C07D215/48;C07D215/50;C07D215/54;C07D217/26;C07D235/06;C07D235/08;C07D235/24;C07D239/26;C07D239/38;C07D241/44;C07D295/12;C07D295/13;C07D295/15;C07D307/79;C07D307/85;C07D401/12;C07K5/02;C07K5/06;C07K5/078;C12N9/99 主分类号 A61K31/17
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