发明名称 |
HMG-COA REDUCTASE INHIBITING SUBSTITUTED PRYIDO (2,3-D) PYRIMIDINES |
摘要 |
New substituted pyrido(2,3-d)pyrimidines of the formula <IMAGE> (I) can be prepared by reduction of corresponding pyrido(2,3-d)-pyrimidines which are substituted by a ketone radical, and subsequent hydrolysis, cyclization or hydrogenation. The new compounds can be used to inhibit HMG-CoA reductase.
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申请公布号 |
US5075311(A) |
申请公布日期 |
1991.12.24 |
申请号 |
US19900460212 |
申请日期 |
1990.01.02 |
申请人 |
BAYER AKTIENGESELLSCHAFT |
发明人 |
HUEBSCH, WALTER;ANGERBAUER, ROLF;FEY, PETER;PHILIPPS, THOMAS;BISCHOFF, HILMAR;PETZINNA, DIETER;SCHMIDT, DELF;THOMAS, GUENTER |
分类号 |
A61K31/505;A61P3/06;A61P9/10;C07D471/04 |
主分类号 |
A61K31/505 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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