发明名称 PROCESS FOR THE PRODUCTION OF N-(PYRROLO/2,3-D/PYRIMIDINE-3-YL-ACYL)-GLUTAMINE-ACID DERIVATIVES
摘要 <p>N-(Acyl)glutamic acid derivatives in which the acyl group is substituted with 4-hydroxypyrrolo[2,3-d]pyrimidin-3-yl group are antineoplastic agents. A typical embodiment is N-[4-(2-{4-hydroxy-6-aminopyrrolo[2,3-d]pyrimidin-3-yl}-ethyl)benzoyl] -L-glutamic acid.</p>
申请公布号 HU908147(D0) 申请公布日期 1991.06.28
申请号 HU19900008147 申请日期 1990.12.10
申请人 THE TRUSTEES OF PRINCETON UNIVERSITY,US 发明人 TAYLOR,EDWARD C.,US;KUHNT,DIETMAR G.,DE;SHIH,CHUAN,US;GRINDEY,GERALD B.,US
分类号 C07D487/04;A61K31/195;A61K31/505;A61K31/519;A61P35/00;A61P35/02;A61P43/00 主分类号 C07D487/04
代理机构 代理人
主权项
地址