发明名称 |
PYRIMIDINE-4,6-DICARBOXYLIC ACID DIAMIDES,PROCESSES FOR THEIR PREPARATION AND THE USE THEREOF,AND PHARMACEUTICALS BASED ON THESE COMPOUNDS |
摘要 |
The invention relates to pyrimidine-4,6-dicarboxamides of the formula I …<IMAGE>… in which R<1> and R<2> have the stated meanings. The compounds according to the invention inhibit proline hydroxylase and lysine hydroxylase and can be used as fibrosuppressants and immunosuppressants. |
申请公布号 |
ZA9007535(B) |
申请公布日期 |
1991.06.26 |
申请号 |
ZA19900007535 |
申请日期 |
1990.09.20 |
申请人 |
HOECHST AKTIENGESELLSCHAFT |
发明人 |
EKKEHARD BAADER;VOLKMAR GUENZLER-PUKALL;MARTIN BICKEL;STEPHAN HENKE |
分类号 |
A61K31/505;A61K31/535;A61P3/00;A61P37/06;C07D239/28;C07D401/14;C07D403/14;C07D409/14;C07D413/14;C07D417/14 |
主分类号 |
A61K31/505 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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