发明名称 |
SLOWLY DISSOCIATING (TIGHT BINDING) DOPAMINE, SEROTONIN OR NOREPINEPHRINE REUPTAKE INHIBITORS AS COCAINE, AMPHETAMINE AND PHENCYCLIDINE ANTAGONISTS |
摘要 |
Methods are disclosed for treating cocaine addiction, acute effects of cocaine, and cocaine craving in mammals using a cocaine antagonist of general formula (I). The methods of treatment can counteract cocaine intoxication and prevent relapse into drug use during and after treatment. Preferably, (1-[2-[bis(4-fluorophenyl)-methoxy]ethyl]-4-[3-phenylpropyl]-piperizine is administered in the range of 0.1 mg to 100 mg per kg body weight per day. |
申请公布号 |
AU6277890(A) |
申请公布日期 |
1991.03.11 |
申请号 |
AU19900062778 |
申请日期 |
1990.08.03 |
申请人 |
UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, UNITED |
发明人 |
RICHARD B. ROTHMAN;AGU PERT;KENNER C. RICE;NIGEL HAMILTON GREIG;AUDREY ALICE REID;HYACINTH CHARLES CHI AKUNNE;ANDRE MELE;ANDREW THURKAUF |
分类号 |
A61K31/495;A61P25/00;A61P25/30;C07D295/08 |
主分类号 |
A61K31/495 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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