发明名称 Process of preparing 2-(imidazolin-2-yl)-nicotinic acid compounds
摘要 The invention relates to processes for the preparation of 6-substituted 2-(imidazolin-2-yl)-nicotinic acid derivatives that are distinguished by excellent herbicidal and plant growth-regulating properties, and to intermediates and processes for the preparation of the intermediates. The derivatives correspond to formula I <IMAGE> (I) in which R1 represents hydrogen or a salt, ester or amide radical, each of R2 and R3, independently of the other, represents C1-C4-alkyl or they together represent a C3-C5-alkylene radical, X represents hydrogen or methyl, Y represents hydrogen, halogen, alkyl, haloalkyl, hydroxyalkyl, alkoxy, alkylthio, phenoxy, nitro, cyano, alkylamino, phenyl, alkenyloxy or alkynyloxy, and Z represents a -CQ1Q2Q3 or -CQ1Q4Q5 radical in which Q1 and Q2 each represents hydrogen or C1-C4-alkyl, Q3 represents C1-C6-alkoxy or phenoxy that is unsubstituted or substituted, or C3-C6-alkenyloxy or C3-C6-alkynyloxy and Q4 and Q5, together with the carbon atom to which they are bonded, represent a cycloalkyl, furyl, pyran, dioxan or dioxolan radical, or Z represents a 5- or 6-membered heterocyclic radical.
申请公布号 US4997947(A) 申请公布日期 1991.03.05
申请号 US19890426901 申请日期 1989.10.24
申请人 CIBA-GEIGY CORPORATION 发明人 SZCZEPANSKI, HENRY;DUERR, DIETER
分类号 A01N43/50;A01N43/90;C07D213/80;C07D401/04;C07D401/14;C07D405/14;C07D409/14;C07D471/04;C07D471/14;C07D491/04;C07D491/048 主分类号 A01N43/50
代理机构 代理人
主权项
地址