发明名称 ANDROGEN DERIVATIVES FOR USE IN THE INHIBITION OF SEX STEROID ACTIVITY
摘要 Methods for treating sex steroid-dependent diseases by inhibiting sex steroid activity include administration of novel compounds which include an androgenic nucleus substituted at a ring carbon with at least one substituent specified herein. Such compounds may function by inhibiting sex steroid synthesis (both estrogen and androgen synthesis) and/or by antagonistically blocking androgen receptors.
申请公布号 WO9100732(A1) 申请公布日期 1991.01.24
申请号 WO1990CA00211 申请日期 1990.07.05
申请人 ENDORECHERCHE INC. 发明人 LABRIE, FERNAND;MERAND, YVES
分类号 A61K31/00;A61K31/565;A61K31/57;A61K31/575;A61K31/58;A61K31/585;A61K31/66;A61K31/695;A61P5/24;C07C235/34;C07D235/18;C07J1/00;C07J7/00;C07J9/00;C07J17/00;C07J21/00;C07J41/00;C07J43/00;C07J51/00;C07J73/00 主分类号 A61K31/00
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