发明名称 |
ANDROGEN DERIVATIVES FOR USE IN THE INHIBITION OF SEX STEROID ACTIVITY |
摘要 |
Methods for treating sex steroid-dependent diseases by inhibiting sex steroid activity include administration of novel compounds which include an androgenic nucleus substituted at a ring carbon with at least one substituent specified herein. Such compounds may function by inhibiting sex steroid synthesis (both estrogen and androgen synthesis) and/or by antagonistically blocking androgen receptors. |
申请公布号 |
WO9100732(A1) |
申请公布日期 |
1991.01.24 |
申请号 |
WO1990CA00211 |
申请日期 |
1990.07.05 |
申请人 |
ENDORECHERCHE INC. |
发明人 |
LABRIE, FERNAND;MERAND, YVES |
分类号 |
A61K31/00;A61K31/565;A61K31/57;A61K31/575;A61K31/58;A61K31/585;A61K31/66;A61K31/695;A61P5/24;C07C235/34;C07D235/18;C07J1/00;C07J7/00;C07J9/00;C07J17/00;C07J21/00;C07J41/00;C07J43/00;C07J51/00;C07J73/00 |
主分类号 |
A61K31/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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