发明名称 ADDITIONSPRODUKTER AF 3,4-DIHYDRO-4-OXO-2H-1,2-BENZOTHIAZIN-3-CARBOXYLSYRE-1,1-DIOXID-ESTERE OG HETEROCYCLISK SUBSTITUEREDE AMINER.
摘要 A novel compound of empirical formula C9H7N2O5SRR<1>Z (I) produced by reacting an ester of the formula <CHEM> with an equimolar amount of an amine of the formula ZNH2 in a reaction inert organic solvent at a temperature of from about 0 to 110 DEG C wherein R is hydrogen benzyl or (C1-C3) alkyl; R<1> is benzyl or (C1-C4) alkyl and Z is benzopyronyl, alkyl substituted benzopyronyl, 2-pyridyl, alkyl substituted-2-pyridyl, 2-thiazolyl, 2-thiazolyl substituted by one or two alkyl group, or 5-alkyl-3-isoxazolyl, each alkyl having from one to four carbon atoms; and a novel process utilizing the compounds of formula (I) as intermediates for production of known anti-inflammatory agents of the formula <CHEM> u
申请公布号 DK158674(C) 申请公布日期 1991.01.21
申请号 DK19880005751 申请日期 1988.10.14
申请人 PFIZER INC. 发明人 KARDYS, JOSEPH ANTHONY
分类号 C07D417/12;A61K;A61K31/54;C07C;C07D;C07D213/73;C07D261/14;C07D277/20;C07D277/40;C07D279/02;C07D513/22;C07G99/00 主分类号 C07D417/12
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