Benzothiazepine derivatives, process for their preparation and thereby obtained intermediates, their use as medicines and compositions containing them.

摘要

Products of the formula (I) :
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in which :
- X = H, halogen, HO, C1-3 alkyl or alkoxy, NO2, amino, mono or dialkylamino, CF3, SCF3, OCF3, - and either Y =
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with R3 and R4 = H or (C1-4) alkyl,
r and s = integers from 0 to 4,
- or Y =
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with r1 = an integer from 1 to 4,
- or R1 and R2 = H, a (C1-4) alkyl optionally substituted by either optionally substituted (C6-12) aryl or optionally mono- or disubstituted amine or form a heterocycle with 5, 6 or 7 members with optionally another heteroatom, as well as their salts,
a process for their preparation and the intermediates thereby obtained, their application as drugs and the compositions containing them.