发明名称 DERIVATIVES OF IMIDAZOLE, THEIR PREPARATION AND UTILISATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE DERIVATIVES
摘要 <p>Derivatives of imidazole corresponding to formula I wherein X1, X2, Y1 and Y2, whether or not identical, can have different significancies, R1 is hydrogen, a methyl or phenyl group, R2 and R3, whether or not identical, represent hydrogen, a hydroxyl, alkyl or alkoxy group, it being possible for R1 and R2 together to represent a carbon-carbon bond, R4 and R5, whether or not identical, being hydrogen or alkyl, and the tautomers and salts of these compounds, also the pharmaceutical compositions containing them. The compounds are endowed with .alpha.2-blocking and/or anticonvulsive activities and are utilisable as therapeutic agents for man.</p>
申请公布号 CA1273942(A) 申请公布日期 1990.09.11
申请号 CA19860500447 申请日期 1986.01.27
申请人 CONTINENTAL PHARMA INC. 发明人 CALDERON, PIEDAD;CORDI, ALEXIS A.;GILLET, CLAUDE L.;GORISSEN, HUGO J.;LAMBELIN, GEORGES E.;ROBA, JOSEPH L.;SNYERS, MICHEL P.;VAN DORSSER, WILLIAM R.
分类号 A61K31/415;A61P1/04;A61P3/04;A61P3/08;A61P7/02;A61P7/10;A61P9/00;A61P9/12;A61P13/02;A61P15/00;A61P25/02;A61P25/04;A61P25/08;A61P25/24;A61P25/26;C07C17/00;C07C45/63;C07C47/24;C07D233/54;C07D233/58;C07D233/62;C07D233/64;C07D233/84;(IPC1-7):C07D233/64 主分类号 A61K31/415
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