发明名称 FOERFARANDE FOER FRAMSTAELLNING AV GRISEOLINSYRADERIVAT.
摘要 Griseolic acid derivatives of formula (I): <IMAGE> (I) wherein A represents: <IMAGE> have enzyme-inhibitory activity, especially against cAMP PDE and cGMP PDE. When formulated as compositions with appropriate carriers or diluents, they may be used for the treatment of a variety of organic disorders and show toxicities less than griseolic acid itself.
申请公布号 FI81357(B) 申请公布日期 1990.06.29
申请号 FI19840004225 申请日期 1984.10.26
申请人 SANKYO COMPANY LIMITED 发明人 KANEKO, MASAKATSU;KIMURA, MISAKO;MUROFUSHI, YOSHINOBU;YAMAZAKI, MITSUO;IWATA, NOBUYOSHI;NAKAGAWA, FUMIO
分类号 C07H19/16;A61K31/70;A61K31/7042;A61K31/7052;A61K31/7076;A61K31/708;A61P5/12;A61P7/02;A61P25/28;A61P35/00;A61P43/00;C07D307/77;C07D405/06;C07D473/00;C07D473/30;C07D493/04;C07H19/02 主分类号 C07H19/16
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