发明名称 3-VINYL- AND 3- ETHINYL-BETA-CARBOLINE DERIVATIVES
摘要 <p>Compounds of formula I <IMAGE> (I) wherein R1 is hydrogen or a protecting group, R2 is -CH=CR24 or -C 3BOND CR4, R4 is hydrogen or halogen, R3 is hydrogen, lower alkyl or lower alkoxyalkyl, RA is, inter alia, hydrogen, OR7, lower alkyl, which optionally is substituted with aryl, lower alkoxy or NR5R6, R5 and R6 can be the same or different and in each case is hydrogen, lower alkyl or together with the nitrogen atom a 5-6 member ring, which can contain another heteroatom, R7 is lower alkyl, optionally substituted aryl or aralkyl, and each compound can contain one or more RA radicals which are not hydrogen, have valuable pharmacological properties.</p>
申请公布号 AU597001(B2) 申请公布日期 1990.05.24
申请号 AU19860063663 申请日期 1986.10.07
申请人 SCHERING A.G. 发明人 DIETER SEIDELMANN;ANDREAS HUTH;RALPH SCHMIECHEN;PROF. DR. RUDOLF WIECHERT;HERBERT SCHNEIDER;DAVID NORMAN STEPHENS
分类号 A61K31/435;A61P25/00;A61P25/08;A61P25/20;C07D471/04;(IPC1-7):C07D471/04;A61K31/44;A61K31/445;A61K31/535 主分类号 A61K31/435
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