发明名称 |
PROCESS FOR PREPARING CEPHALOSPORIN DERIVATIVES |
摘要 |
Cephalosporin derivs. of fromula (I) are prepd. by reacting a cpd. of formula (II) with a cpd. of formula (III). In the formulas, X is halogen; A is carbonic acid -protecting gp.; R1 is amino-protecting gp.; R is C1-6 alkyl; asterisk indicates (R), (S) or (RS)-form; n is 0 or 1; n' is 0-3; n2 is 0-3. (I) are useful as antibiotics having a high bactericidal activity.
|
申请公布号 |
KR900003563(B1) |
申请公布日期 |
1990.05.21 |
申请号 |
KR19860010043 |
申请日期 |
1986.11.27 |
申请人 |
MEIJI SEIKA KAISHA |
发明人 |
SHIBAHARA SEIJI;OKONOKI TSUNEO;MURAI YASUSHI;KUTO TOSHIAKI;YOSHIDA TAKASHI;NISHIHATA KEN |
分类号 |
A61K31/545;A61K31/546;A61P31/04;C07D501/00;C07D501/36;(IPC1-7):C07D501/36 |
主分类号 |
A61K31/545 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|