发明名称 1,4-diazepine derivative and its pharmaceutical use.
摘要 <p>A triazolo-1,4-di-azepine compound of the below given formula and a pharmacologically acceptable salt thereof are disclosed and useful in the pharmaceutical field, especially to allergic diseases. &lt;CHEM&gt; in which R1 and R2 are hydrogen or an alkyl, R3 is hydrogen or a halogen, R4 is hydrogen or an alkyl, X is -OCO-, -NHCO-, -CO- or others and Y is a cycloalkyl, a cycloalkylalkyl, an alkynyl or others.</p>
申请公布号 EP0367110(A1) 申请公布日期 1990.05.09
申请号 EP19890119910 申请日期 1989.10.26
申请人 EISAI CO., LTD. 发明人 OKANO, KAZUO;MIYAZAWA, SHUHEI;CLARK, RICHARD STEPHEN JOHN;ABE, SHINYA;KAWAHARA, TETSUYA;SHIMOMURA, NAOYUKI;ASANO, OSAMU;YOSHIMURA, HIROYUKI;MIYAMOTO, MITSUAKI;SAKUMA, YOSHINORI;MURAMOTO, KENZO;OBAISHI, HIROSHI;HARADA, KOUKICHI;TSUNODA, HAJIME;KATAYAMA, SATOSHI;YAMADA, KOUJI;SOUDA, SHIGERU;MACHIDA, YOSHIMASA;KATAYAMA, KOUICHI
分类号 C07D495/04;A61K31/55;A61K31/675;A61P11/00;A61P11/08;A61P37/08;C07D495/14;C07D495/22;C07F9/6561 主分类号 C07D495/04
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