发明名称 |
PROCESS FOR PREPARATION OF MEVALONOLACTONES CONTAINING PYRAZOLOPYRIDINE RING AND OF INTERMEDIERS THEREOF AND FOR MANUFACTURING THE PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS |
摘要 |
The present invention relates to compounds of the formula: <CHEM> where Y is -CH2-, -CH2CH2-, -CH=CH-, -CH2-CH=CH-, -CH=CH-CH2-, -C(CH3)=CH- or -CH=C(CH3); Z is -Q-CH2WCH2-CO2R<1><2>, <CHEM> (wherein Q is -C(O)-, -C(OR<1><3>)2- or -CH(OH)-; W is -C(O)-, -C(OR<1><3>)2- or -C(R<1><1>)(OH)-; and their pharmaceutical uses as anti-hyperlipidemic, hypolipoproteinemic and anti-atherosclerotic agents. |
申请公布号 |
HU892751(D0) |
申请公布日期 |
1990.03.28 |
申请号 |
HU19890002751 |
申请日期 |
1989.04.19 |
申请人 |
NISSAN CHEMICAL INDUSTRIES LTD.,JP |
发明人 |
FUJIKAWA,YOSHIHIRO,JP;SUZUKI,MIKO,JP;IWASAKI,HIROSHI,JP;SAKASHITA,MITSUAKI,JP;KITAHARA,MASAKI,JP |
分类号 |
A61K31/435;A61P3/06;A61P9/10;C07D471/04;C07F7/18 |
主分类号 |
A61K31/435 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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