发明名称 NEW BICYCLIC COMPOUNDS,PROCESS FOR PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME
摘要 A bicyclic compound of the following formula : <CHEM> wherein A is @C=O or @CHOH, R<1> is aryl which may have cyano or carbamoyl, or heterocyclic group which may have lower alkyl, R<2> is hydrogen or lower alkyl, R<3> is lower alkyl, X is hydrogen, halogen, hydroxy or lower alkyl, m is an integer 1 or 2, and n is an integer 1 to 4, and pharmaceutically acceptable salts thereof, and processes for their preparation and pharmaceutical compositions comprising them.
申请公布号 PH24176(A) 申请公布日期 1990.03.22
申请号 PH19930000367 申请日期 1988.04.13
申请人 FUJISAWA PHARMACEUTICAL CO.,LTD. 发明人 TERUO OKU;YOSHIO KAWAI;HIROSHI KAYAKIRI;KAZUYOSHI KURATANI;MASASHI HASHIMOTO
分类号 C12N9/99;A61K31/085;A61K31/12;A61K31/165;A61K31/275;A61K31/33;A61K31/415;A61K31/4184;A61K31/425;A61K31/428;A61K31/44;A61K31/4409;A61K31/4418;A61K31/47;A61P1/00;A61P1/16;A61P9/08;A61P9/10;A61P13/02;A61P15/00;A61P29/00;A61P37/08;A61P43/00;C07C41/00;C07C41/01;C07C41/26;C07C43/23;C07C45/00;C07C45/67;C07C45/68;C07C46/00;C07C49/747;C07C49/755;C07C50/12;C07C67/00;C07C231/00;C07C231/06;C07C231/12;C07C235/20;C07C235/42;C07C253/00;C07C253/30;C07C255/32;C07C255/52;C07C255/54;C07D213/30;C07D213/64;C07D215/14;C07D215/20;C07D215/26;C07D231/12;C07D235/08;C07D235/12;C07D237/08;C07D239/26;C07D277/64;C07D277/68;C07D521/00;C07F7/18 主分类号 C12N9/99
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