发明名称 |
1-4-DIAZA-PHENOTHIAZINE ANALOGOUS COMPOUNDS AS 5- LIPOXYGENASE INHIBITORS |
摘要 |
<p>16959Y TITLE OF THE INVENTION 1,4-DIAZA-PHENOTHIAZINE ANALOGOUS COMPOUNDS AS 5-LIPOXYGENASE INHIBITORS Compounds of the Formula I: I are inhibitors of the mammalian 5-lipoxygenase enzyme system of the arachidonic acid cascade. As such, these compounds are useful therapeutic agents for treating allergic conditions, asthma, cardiovascular disorders and inflammation.</p> |
申请公布号 |
CA1261834(A) |
申请公布日期 |
1989.09.26 |
申请号 |
CA19840466743 |
申请日期 |
1984.10.31 |
申请人 |
MERCH FROSST CANADA, INC. |
发明人 |
ATKINSON, JOSEPH;BELANGER, PATRICE C.;GUINDON, YVAN;ROKACH, JOSHUA |
分类号 |
A61K31/495;A61K31/535;A61K31/54;A61P11/00;A61P43/00;C07D241/18;C07D487/04;C07D498/04;C07D513/04;C07D513/16;(IPC1-7):C07D513/04 |
主分类号 |
A61K31/495 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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