| 摘要 |
<p>A compound having the formula K-His-Trp-Ser-Tyr-M-Q-Arg-Pro-T, wherein K is N-Acetyl-Sarconsine or pGlu: is D-Phe, D-Trp, D-.beta. -Nap.hthylalanine, or D-4-X-Phe, wherein X is OH, F, Cl, Br, or Me: Q is Leu, Phe, 4-X-Phe, Trp, or .beta.-Naphthylamine (wherein X is OH, F, Cl, Br, or Me), or an N-Me-derivative thersof: and T is Gly-NH2, NHCH3, NHCH2CH3, or NHCH2CH2CH3; provided that, when Q is Leu or N-Me-Leu, K cannot be pGlu: or a phar~aceutically acceptable salt thereof.</p> |
