发明名称 Phosphinylcycloalkylcarbonyl and phosphinylcycloalkenylcarbonyl dipeptides
摘要 Compounds of the formula <IMAGE> and their pharmaceutically acceptable salts wherein Z completes a cycloalkyl ring, a substituted cycloalkyl ring, a cycloalkenyl ring, a substituted cycloalkenyl ring or a saturated heteroalkyl ring; R2 is lower alkyl, aralkyl or aminoalkyl and X is an amino or imino acid. The compounds possess angiotensin converting enzyme inhibition activity.
申请公布号 US4849525(A) 申请公布日期 1989.07.18
申请号 US19870098651 申请日期 1987.09.21
申请人 E. R. SQUIBB & SONS, INC. 发明人 WELLER, III, HAROLD N.;GORDON, ERIC M.
分类号 A61K38/55;A61K31/675;A61K38/00;A61P9/12;A61P43/00;C07K5/06;C07K5/08;C07K14/81;C12N9/99 主分类号 A61K38/55
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