发明名称 |
Oligopeptide prodrugs |
摘要 |
Prodrugs are described whose structures have a oligopeptide chain which is substituted by a nucleophilic chemotherapeutic residue at the alpha -position. The products have increased cell membrane permeability and beneficial physico-chemical properties.
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申请公布号 |
US4454065(A) |
申请公布日期 |
1984.06.12 |
申请号 |
US19830507326 |
申请日期 |
1983.06.23 |
申请人 |
SMITHKLINE BECKMAN CORPORATION |
发明人 |
GILVARG, CHARLES;KINGSBURY, WILLIAM D. |
分类号 |
A61K38/00;C07K5/06;C07K5/065;C07K5/083;C07K7/06;(IPC1-7):C07C103/52 |
主分类号 |
A61K38/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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