发明名称 |
10-aryl-1,8-dihydroxy-9-anthrones and their esters, process for preparing same, and use of same in human and veterinary medicine and in cosmetics |
摘要 |
Mono, di and tri-esters of 1,8-dihydroxy-10-phenyl-9-anthrone or -9-anthranol have the formula <IMAGE> (I) wherein p is 0 or 1, (a) when p=0, t=1 and R2 represents hydrogen or -COR3, (b) when p=1, t=0 and R1 and R2 each independently represent hydrogen or -COR3, R3 represents linear or branched alkyl having 1-17 carbon atoms, cycloalkyl, phenyl or phenyl substituted by lower alkyl, lower alkoxy, halogen, a nitro function, -CF3 or a hydroxyl function, and mixtures of said esters. These esters are prepared by reacting 1,8-dihydroxy-10-phenyl-9-anthrone with an activated form of an acid. The esters are useful in human or veterinary medicine and in cosmetic compositions.
|
申请公布号 |
US4843097(A) |
申请公布日期 |
1989.06.27 |
申请号 |
US19880176974 |
申请日期 |
1988.04.04 |
申请人 |
GROUPEMENT D'INTERET ECONOMIQUE DIT: CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES C.I.R.D. |
发明人 |
SHROOT, BRAHAM;LANG, GERARD;MAIGNAN, JEAN;RESTLE, SERGE;HENSBY, CHRISTOPHER;COLIN, MICHEL |
分类号 |
A61K8/37;A61K31/215;A61Q5/00;A61Q7/00;A61Q19/00;C07D277/24;C07D333/22;C07D333/24 |
主分类号 |
A61K8/37 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|