发明名称 FOERFARANDE OCH MELLANPRODUKTER FOER FRAMSTAELLNING AV BENZOTIAZINKARBOXAMIDER.
摘要 A novel compound of empirical formula C9H7N2O5SRR<1>Z (I) produced by reacting an ester of the formula <CHEM> with an equimolar amount of an amine of the formula ZNH2 in a reaction inert organic solvent at a temperature of from about 0 to 110 DEG C wherein R is hydrogen benzyl or (C1-C3) alkyl; R<1> is benzyl or (C1-C4) alkyl and Z is benzopyronyl, alkyl substituted benzopyronyl, 2-pyridyl, alkyl substituted-2-pyridyl, 2-thiazolyl, 2-thiazolyl substituted by one or two alkyl group, or 5-alkyl-3-isoxazolyl, each alkyl having from one to four carbon atoms; and a novel process utilizing the compounds of formula (I) as intermediates for production of known anti-inflammatory agents of the formula <CHEM> u
申请公布号 FI77657(C) 申请公布日期 1989.04.10
申请号 FI19820002697 申请日期 1982.08.02
申请人 PFIZER INC., 发明人 KARDYS,JOSEPH ANTHONY
分类号 C07D277/20;A61K31/54;C07D213/73;C07D261/14;C07D277/40;C07D279/02;C07D417/12;C07D513/22;C07G99/00;(IPC1-7):C07D279/02 主分类号 C07D277/20
代理机构 代理人
主权项
地址