发明名称 DERIVATI DI INDOLO,PROCEDIMENTI PER PREPARARLI E COMPOSIZIONI FARMACEUTICHE CHE LI CONTENGONO PER IL TRATTAMENTO DI EMICRANIA
摘要 Indole derivs. of formula (I) and their salts are new. R1 = halogen, 1-3C alkoxy, R6R7NCO(CH2)p, R6CONH(CH2)p, R6R7NSO2 (CH2)p or R8SO2NH (CH2)p; R6, R7 = H or 1-3C alkyl; R8 = 1-3C alkyl; p = 0 or 1; R2 = H or 1-3C alkyl, R3 = H or 1-3C alkyl, R4, R5 = H, 1-3C alkyl or 2-propenyl; A = CO or SO, n = 2-5; m = 0-4. - Also new are cpds. of formula (II) used in the prepn. of (I).
申请公布号 IT1205849(B) 申请公布日期 1989.03.31
申请号 IT19870047507 申请日期 1987.01.08
申请人 GLAXO GROUP LTD. 发明人 MILLS KEITH;ELDRED COLIN DAVID;OXFORD ALEXANDER WILLIAM;COATES IAN HAROLD;BAYS DAVID EDMUND;WEBB COLIN FREDERICK;DOWLE MICHAEL DENNIS
分类号 C07D209/14;A61K31/40;A61K31/403;A61K31/404;A61K31/405;A61P9/00;A61P25/04;C07D209/16 主分类号 C07D209/14
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