发明名称 4H-3,1-BENZOXAZINE DERIVATIVE, PRODUCTION THEREOF AND AGRICULTURAL AND HORTICULTURAL FUNGICIDE CONTAINING SAID DERIVATIVE
摘要 NEW MATERIAL:A 4H-3,1-benzoxazine derivative shown by formula I (Y is halogen or lower alkyl; n is 0-2; two Y may be the same or different when n is 2 in Yn; R is H, alkyloxy, alkynyloxy, alkylthio or alkenylthio). EXAMPLE:4-(4-Chlorophenyl)-4-isopropyloxy-2-(4-pyridyl)-4H-3,1-benzoxa zine. USE:Useful as an agriculatural and horticultural fungicide applicable to various pathogenic germs such as Phycomycetes and Ascomycetes, showing excellent effects especially on powdery mildew, rust, downy mildew and dampling-off useful plants. PREPARATION:A benzophenone derivative shown by formula II is reacted with a halogenating agent to give a reaction product, which is reacted with a corresponding alcohol or thiol to give a compound shown by formula I.
申请公布号 JPS63264480(A) 申请公布日期 1988.11.01
申请号 JP19880086913 申请日期 1988.04.08
申请人 CHUGAI PHARMACEUT CO LTD 发明人 SUGIYAMA HIROSHI;HOSODA KEIZO;KUMAGAI YOSHIKAZU;TAKEUCHI MASAKI;OKADA MASANORI
分类号 C07D413/04;A01N43/86 主分类号 C07D413/04
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