发明名称 |
3-oxadiazole and 3-carboxylic acid beta-carboline derivatives, and their use as psychotropic agents |
摘要 |
Compounds of formula I <IMAGE> (I) wherein X is COOR3 or an oxadiazolyl radical of the formula or R2 is H, lower alkyl or cycloalkyl, R3 is lower alkyl, R4 is hydrogen, lower alkyl or lower alkoxyalkyl, RA is -CHR1-Z-R5, Z is sulfur or oxygen, R1 is lower alkyl or optionally substituted phenyl, and R5 is hydrogen, phenyl or optionally substituted lower alkyl, and wherein each compound can contain 1 or 2 RA radicals have valuable pharmacological properties.
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申请公布号 |
US4778800(A) |
申请公布日期 |
1988.10.18 |
申请号 |
US19860929866 |
申请日期 |
1986.11.13 |
申请人 |
SCHERING AKTIENGESELLSCHAFT |
发明人 |
HUTH, ANDREAS;SCHMIECHEN, RALPH;STEPHENS, DAVID N.;ENGELSTOFT, MOGENS;WAETJEN, FRANK;HANSEN, JOHN B.;JENSEN, LEIF H. |
分类号 |
A61K31/435;A61P25/08;A61P25/20;C07D471/04;(IPC1-7):A61K31/40 |
主分类号 |
A61K31/435 |
代理机构 |
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地址 |
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