发明名称 ANTIBIOTIC BETA-LACTAMS CONTAINING A PYRIDONE CARBOXYLIC ACID OR ACID DERIVATIVE
摘要 PCT No. PCT/US88/00206 Sec. 371 Date Aug. 24, 1989 Sec. 102(e) Date Aug. 24, 1989 PCT Filed Feb. 1, 1988 PCT Pub. No. WO88/06587 PCT Pub. Date Sep. 7, 1988.This invention presents novel 2-azetidinone compounds of the formula <IMAGE> +TR <IMAGE> wherein R80 is -CO2R5 or -CONR6R7; wherein R5 is hydrogen or (C1-C4) alkyl; and wherein R6 and R7 are the same or different and are hydrogen, (C1-C4 alkyl), or -OH with the proviso that when R6 is -OH, R7 is other than -OH. These compounds are useful as antibacterial agents to eradicate or control susceptible microbes. Intermediates and processes for making these compounds are also disclosed.
申请公布号 AU1180288(A) 申请公布日期 1988.09.26
申请号 AU19880011802 申请日期 1988.02.01
申请人 THE UPJOHN COMPANY 发明人 KYOUNG S. KIM
分类号 C07D205/085;A61K31/397;A61K31/44;A61K31/4418;A61K31/4427;A61P31/04;C07D213/80;C07D401/12;C07D401/14;C07D417/12;C07D417/14 主分类号 C07D205/085
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