发明名称 NYA -LAKTAMASINHIBITORFOERENINGAR.
摘要 The present invention relates to hitherto unknown compounds of the general formula I: <IMAGE> I in which R1 stands for a phenyl, 4-hydroxyphenyl, 1,4-cyclohexadienyl or a 3-thienyl group; R2 represents a primary amino or a carboxy group; R3 is a hydrogen atom, or a lower alkyl, aryl or aralkyl radical, and A stands for a radical of a beta -lactamase inhibitor containing a beta -lactam ring as well as a carboxy group, A being connected via the carboxy group. The present invention provides new compounds useful in the treatment of bacterial infections. The new compounds are in particular strongly active against beta -lactamase producing bacteria.
申请公布号 FI76807(B) 申请公布日期 1988.08.31
申请号 FI19870000555 申请日期 1987.02.11
申请人 LEO PHARMACEUTICAL PRODUCTS LTD. A/S/(LOEVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) 发明人 GODTFREDSEN, WAGN OLE;VON DAEHNE, WELF
分类号 C07D;C07D498/04;C07D499/00;C07D499/21;C07D499/32;C07D499/64;C07D499/68;C07D499/72;C07D499/74;C07D503/00;C07D519/00;(IPC1-7):C07D499/00 主分类号 C07D
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